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Drug-like Properties: Concepts, Structure Design and Methods from ADME to Toxicity Optimization


This book explains the drug discovery process and how property based design can increase the success rate of bringing compounds to market. Drug-like ...

  • CodeCallNoLokasiKetersediaan
    01021080500253Tersedia
  • Perpustakaan
    Fakultas Farmasi
    Judul Seri
    -
    No. Panggil
    615.1-1 Ker D
    Penerbit Academic Press : USA.,
    Deskripsi Fisik
    Ed.1-Cet.1. xix, 526 hal. Ilus. ; 26,5 cm Index. H
    Bahasa
    Indonesia
    ISBN/ISSN
    9.78012E+12
    Klasifikasi
    615.1-1 Ker D
    Tipe Isi
    -
    Tipe Media
    -
    Tipe Pembawa
    -
    Edisi
    NULL
    Subyek
    Info Detil Spesifik
    -
    Pernyataan Tanggungjawab
  • This book explains the drug discovery process and how property based design can increase the success rate of bringing compounds to market. Drug-like properties, such as solubility, permeability, and metabolism, are examined as the fundamental determinants of how drugs behave in vivo. The concepts of pharmacokinetics are discussed with a minimum of mathematical equations, placing emphasis on their practical applications to drug discovery projects. The book has 5 part. Part 1 about introductory concepts. Part 2 about physicochemical properties. Part 2 about physicochemical properties. Part 3 about disposition, metabolism, and safety. Part 4 about methods. Part 5 about specific topics.
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